Assistant Professor of Biochemistry
Department of Chemistry and Biochemistry
Contact Information:
Email: Bouley.8@osu.edu
Office: Marion Science and Engineering (MSE) 110G
Education and Training:
2016–2019 Postdoctoral Research Fellow
University of Michigan, Life Sciences Institute and Department of Pharmacology
2016 Ph.D. Organic Chemistry
University of Notre Dame, Department of Chemistry and Biochemistry
Thesis Title: Development of New Antibacterial Agents for the Treatment of Methicillin-Resistant Staphylococcus aureus
2010 B.S. Chemistry
Grand Valley State University, Department of Chemistry
Honors and Awards:
2017 Molecular Pharmacology Highlighted Trainee Author
2017 Young Chemist Society CIBA Young Scientist Travel Award
2017 Robert M. Scarborough Graduate Award for Excellence in Medicinal Chemistry
2017 The Eli J. and Helen Shaheen Graduate School Award in Science
- Recognizes one graduate student from each division of the Graduate School
2016 The Dow Chemical Outstanding Graduate Student Award
- Recognizes one graduate student from the department
2015 Baxter Young Investigator Award (Second Tier Winner)
2014 Oral Presentation Award, Chemistry-Biochemistry-Biology Interface Symposium
Publications:
- Rasheed S*, Bouley RA, Yoder RJ, Petreaca RC. In silico analysis of driver PRMT5 mutations in cancer cells. J. Mol. Sci. (2023) 24, 6042. PMID:37047013
- Hardison KL*, Hawk TM*, Bouley RA, Petreaca RC. KAT5 histone acetyltransferase mutations in cancer cells. microPublication Biology. (2022) Doi: 10.17912/micropub.biology.000676
- Hamid AN*, Frank LE*, Bouley RA, Petreaca RC. Pan-Cancer Analysis of Co-Occurring Mutations in RAD52 and BRCA1-BRCA2-PALB2 Axis in Human Cancers. PLOS One (2022) 13, 4299. PMID: 34503108.
- Pappula AL*, Gibson LM*, Bouley RA, Petreaca RC. In silico analysis of a SLC6A4 G100V mutation in lung cancers. microPublication Biology. (2022) Doi: 10.17912/micropub.biology.000645
- Bouley R. Redesigning a 1-Semester Biochemistry Class Using In-Class Activities to Achieve High Student Engagement. Chem. Ed. (2022) 99, 293-2949. Doi: 10.1021/acs.jchemed.2c00184
- Martinez-Caballero S, Mahasenan KV, Kim C, Molina R, Feltzer R, Lee M, Bouley R, Hesek D, Fisher JF, Chang M, Mobashery S, Hermoso JA. Integrative Structural Biology of the Essential Penicillin-Binding Protein-1, a Component of the Divisome of Staphylococcus aureus. Struct. Biotech. J. (2021) 19, 5392. PMID: 34667534
- Pappula AL*, Rasheed S*, Mirzaei M, Petreaca RC, Bouley RA. A Genome-Wide Profiling of Glioma Patients with an IDH1 Mutation Using the Catalogue of Somatic Mutations in Cancer Database. Cancers (2021) 13, 4299. PMID: 3450108
- Rowlands R, Chen Q, Bouley R, Avramova L, Tesmer JJG, White A. Generation of Highly Selective, Potent, and Covalent G Protein-Coupled Receptor Kinase 5 Inhibitors. Med. Chem. (2020)
- Holub AS, Bouley RA, Petreaca RC, Husbands AY. Identifying Cancer-Relevant Mutations in the DLC START Domain Using Evolutionary and Structure-Function Analysis. J. Mol. Sci. (2020) 21, 8175.
- Bouley RA, Weinberg ZY, Waldschmidt HV, Yen YC, Larsen SD, Puthenveedu MA, Tesmer JJG. Pharm. (2020) 97, 392-401. PMID: 32234810
- Rowlands R, Cato MC, Waldschmidt HV, Bouley R, Chen Q, Avramova L, Larsen SD, Tesmer JJG, White A. Structure-Based Design of Selective, Covalent G Protein-Coupled Receptor Kinase 5 Inhibitors. ACS Med. Chem. Lett. (2019) 10, 1628-1634. PMID: 31857838
- Bouley R, Hinkovska-Galcheva V, Shayman JA, Tesmer JJG. Structural basis of lysosomal phospholipase A2 inhibition by Zn2+. Biochemistry (2019). PMID: 30830753
- Janardhanan J, Bouley R, Martinez-caballero S, Peng Z, Batuecas-Mordillo M, Meisel J, Ding D, Schroeder VA, Wolter Wa, Mahasenan K, Hermoso JA, Mobashery S, Chang M. The quinazolinone allosteric inhibitor of PBP2a synergizes with piperacillin and tazobactam against methicillin-resistant Staphylococcus aureus. Agents Chemother. (2019). PMID: 30858202
- Hinkovska-Galcheva V, Kelly RJ, Manthei KA, Bouley R, Yuan W, Schwendeman A, Tesmer JJG, Shayman JA. Determinants of pH profile and acyl chain selectivity in lysosomal phospholipase A2. Lipid Res. (2018) 59, 1205-1218. PMID: 29724779
- Waldschmidt HV, Bouley R, Kirchoff PD, Tesmer JJG, Larsen SD. Utilizing a Structure-Based Docking Approach to Develop Potent G Protein-Coupled Receptor Kinase (GRK) 2 and 5 Inhibitors. Med. Chem. Lett. (2018) 28, 1507-1515. PMID: 29627263
- Bouley R, Waldschmidt HV, Cato MC, Cannavo A, Song J, Cheung JY, Yao X, Koch WJ, Larsen SD, Tesmer JJG. Structural Determinants Influencing the Potency and Selectivity of Indazole-Paroxetine Hybrid G Protein-Coupled Receptor Kinase 2 Inhibitors. Pharm. (2017) 92, 707-717. PMID: 29070696
- Mahasenan KV, Molina R, Bouley R, Batuecas MT, Fisher JF, Hermoso JA, Chang M, Mobashery, S. Conformational dynamics in Penicillin-binding protein 2a of Methi-cillin-resistant Staphylococcus aureus, allosteric communication network and enablement of catalysis. Am. Chem. Soc. (2017) 139, 2102-2110. PMID: 28099001
- Bouley R, Ding D, Peng Z, Bastian M, Lastochkin E, Song W, Suckow MA, Schroeder VA, Wolter WR, Mobashery S, Chang M. Structure-Activity Relationship for the 4(3H)-Quinazolinone Antibacterials. Med. Chem.(2016) 59, 5011-5021. PMID: 27088777
- Gonzales PR, Pesesky MW, Bouley R, Ballard A, Suckow MA, Biddy BA, Wolter WR, Schroeder VA, Burnham CD, Mobashery S, Chang M, Dantas G. Synergistic, collaterally-sensitive β-lactam combinations suppress resistance in MRSA. Chem. Biol. (2015) 11, 855-861. PMID: 26268589
- Wang H, Lee M, Peng Z, Blazquez B, Lastochkin E, Kumarasiri M, Bouley R, Chang M, Mobashery S. Synthesis and Evaluation of 1,2,4-Triazolo[1,5-a]pyrimidines as Antibacterial Agents Against Enterococcus faecium. Med. Chem. (2015) 58, 4194-4203. PMID: 25923368
- Bouley R, Kumarasiri M, Peng Z, Otero LH, Song W, Suckow MA, Schroeder VA, Wolter WA, Lastochkin E, Antunes NT, Pi H, Vakulenko S, Hermoso JA, Chang M, Mobashery S. Discovery of Antibiotic (E)-3-(3-Carboxyphenyl)-2-(4-cyanostyryl)quinazolin-4(3H)-one. J. Am. Chem. Soc. (2015) 137, 1738-1741. PMID: 25629446
- Testero S, Bouley R, Fisher J, Chang M, Mobashery S. Exploration of Mild Copper-Mediated Coupling of Organotrifluoroborates in the Synthesis of Thiirane-Based Inhibitors of Matrixmetalloproteinases. Med. Chem. Lett. (2011) 21, 2675-2678. PMID: 21256011